Fluorinated pyrazole acids are agonists of the high affinity niacin receptor GPR109a
Philip J. Skinnera, Martin C. Cherriera, Peter J. Webba, Young-Jun Shina, Tawfik Gharbaouia, Andrew Lindstroma,
Vu Honga, Susan Y. Tamuraa, Huong T. Dangb,Cameron C. Prideb, Ruoping Chenb, Jeremy G. Richmanb,
Daniel T. Connollyb, Graeme Semplea
Bioorganic & Medicinal Chemistry Letters, Volume 17, Issue 20, 15 October 2007, Pages 5620–5623
- DOI:
http://dx.doi.org/10.1016/j.bmcl.2007.07.101