+++thanks_2 articles from ACS

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1. Design, Synthesis, and Biological Evaluation of Novel Conformationally Constrained Inhibitors Targeting EGFR
Jianwei Wu †, Wenteng Chen †, Guangxin Xia ‡, Jing Zhang ‡, Jiaan Shao †, Biqin Tan §, Chunchun Zhang ‡, Wanwan Yu †, Qinjie Weng §, Haiyan Liu ‡, Miao Hu †, Hailin Deng ‡, Yu Hao ‡, Jingkang Shen *‡, and Yongping Yu

ACS Med. Chem. Lett., 2013, 4 (10), pp 974–978

DOI:

http://dx.doi.org/10.1021/ml4002437

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http://pubs.acs.org/doi/abs/10.1021%2Fml4002437

2. Structure-Based Approach for the Discovery of Pyrrolo[3,2-d]pyrimidine-Based EGFR T790M/L858R Mutant Inhibitors
Satoshi Sogabe *, Youichi Kawakita , Shigeru Igaki , Hidehisa Iwata , Hiroshi Miki , Douglas R. Cary , Terufumi Takagi , Shinji Takagi , Yoshikazu Ohta , and Tomoyasu Ishikawa *
ACS Med. Chem. Lett., 2013, 4 (2), pp 201–205

DOI:

http://dx.doi.org/10.1021/ml300327z

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http://pubs.acs.org/doi/abs/10.1021/ml300327z?journalCode=amclct&quickLinkVolume=4&quickLinkPage=201&selectedTab=citation&volume=4