Synthesis of highly potent and selective hetaryl ureas as integrin αVβ3-Receptor antagonists
Udo E. W. Lange, Gisela Backfisch, Jürgen Delzer, Hervé Geneste, Claudia Graef, Wilfried Hornberger, Andreas Kling, Arnulf Lauterbach, Thomas Subkowski, Christian Zechel
Bioorganic & Medicinal Chemistry Letters, Volume 12, Issue 10, 20 May 2002, Pages 1379-1382
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http://dx.doi.org/10.1016/S0960-894X(02)00161-0