Efficacious and Orally Bioavailable Thrombin Inhibitors Based on a 2,5-Thienylamidine at the P1 Position: Discovery of N-Carboxymethyl-D-diphenylalanyl-L-prolyl[(5-amidino-2-thienyl)methyl]amide
Koo Lee, Cheol Won Park, Won-Hyuk Jung, Hee Dong Park, Sun Hwa Lee, Kyung Ha Chung, Su Kyung Park, O Hwan Kwon, Myunggyun Kang, Doo-Hee Park, Sang Koo Lee, Eunice E. Kim, Suk Kyoon Yoon, and Aeri Kim
J. Med. Chem.; 2003; 46(17) pp 3612 - 3622; (Article) DOI: 10.1021/jm030025j
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http//dx.doi.org/10.1021/jm030025j