1. Timo Heinrich, Henning Böttcher, Rolf Gericke et al.
"Synthesis and Structure−Activity Relationship in a Class of Indolebutylpiperazines as Dual 5-HT1A Receptor Agonists and Serotonin Reuptake Inhibitors"
J. Med. Chem., 2004, Vol. 47, Issue 19, pp. 4684–4692.
- DOI:
http://dx.doi.org/10.1021/jm040793q
"Indolebutylamines as Selective 5-HT1A Agonists"
J. Med. Chem., 2004, Vol. 47, Issue 19, pp. 4677–4683.
- DOI:
http://dx.doi.org/10.1021/jm040792y
"3-(4-Piperidinylalkyl)indoles, selective inhibitors of neuronal 5-hydroxytryptamine uptake"
J. Med. Chem., 1980, Vol. 23, Issue 12, pp. 1306–1310.
- DOI:
http://dx.doi.org/10.1021/jm00186a005
"Synthesis of New Arylpiperazinylalkylthiobenzimidazole, Benzothiazole, or Benzoxazole Derivatives as Potent and Selective 5-HT1A Serotonin Receptor
Ligands"
J. Med. Chem., 2008, Vol. 51, Issue 15, pp. 4529–4538.
- DOI:
http://dx.doi.org/10.1021/jm800176x
"Discovery of a Novel 5-HT3 Antagonist/5-HT1A Agonist 3-Amino-5,6,7,8-tetrahydro-2-{4-[4-(quinolin-2-yl)piperazin-1-yl]butyl}quinazolin-4(3H)-one (TZB-
30878) as an Orally Bioavailable Agent for Irritable Bowel Syndrome"
J. Med. Chem., 2010, Vol. 53, Issue 21, pp. 7549–7563.
- DOI:
http://dx.doi.org/10.1021/jm1002292
"New 1-Aryl-3-(4-arylpiperazin-1-yl)propane Derivatives, with Dual Action at 5-HT1A Serotonin Receptors and Serotonin Transporter, as a New Class of
Antidepressants"
J. Med. Chem., 2001, Vol. 44, Issue 3, pp. 418–428.
- DOI:
http://dx.doi.org/10.1021/jm001059j
"Structure−Affinity Relationship Study on N-(1,2,3,4-Tetrahydronaphthalen-1-yl)-4-Aryl-1-Piperazinealkylamides, a New Class of 5-Hydroxytryptamine7
Receptor Agents"
J. Med. Chem., 2004, Vol. 47, Issue 26, pp. 6616–6624.
- DOI:
http://dx.doi.org/10.1021/jm049702f
"Receptor-Based Pharmacophores for Serotonin 5-HT7R Antagonists Implications to Selectivity"
J. Med. Chem., 2006, Vol. 49, Issue 23, pp. 6732–6741.
- DOI:
http://dx.doi.org/10.1021/jm060300c