+++Elsevier

[Ligand]

1. Novel 3-aroylpyrazolo[5,1-c][1,2,4]benzotriazine 5-oxides 8-substituted, ligands at GABAA/benzodiazepine receptor complex: Synthesis, pharmacological and molecular modeling studies
Gabriella Guerrinia, Giovanna Ciciania, Giovanni Cambia, Fabrizio Brunia, Silvia Selleria, Fabrizio Melanib, Marina Montalic, Claudia Martinic, Carla Ghelardinid, Monica Norcinid and Annarella Costanzo
Bioorganic & Medicinal Chemistry
Article in Press

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http://dx.doi.org/10.1016/j.bmc.2008.02.058

2. 3D and quantum QSAR of non-benzodiazepine compounds
F.A. Pashaa, M. Muddassara, Seung Joo Choa, Kaleem Ahmadb and Yakub Beg
European Journal of Medicinal Chemistry
Article in Press,

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http://dx.doi.org/10.1016/j.ejmech.2008.01.030

3. In Vivo Characterization and Dynamic Receptor Occupancy Imaging of TPA023B, an α2/α3/α5 Subtype Selective γ-Aminobutyric Acid–A Partial Agonist
Koen Van Laerea, Guy Bormansc, Sandra M. Sanabria-Bohórquezf, Tjibbe de Grootc, Patrick Duponta, Inge De Lepeleired, Jan de Hoonb, Luc Mortelmansa, Richard J. Hargreavesf, John R. Atacke, g and H. Donald Burns
Biological Psychiatry
Article in Press,

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http://dx.doi.org/10.1016/j.biopsych.2008.01.021

4. QSAR modeling of the interaction of flavonoids with GABA(A) receptor
Pablo R. Duchowicza, Martín G. Vitalea, Eduardo A. Castroa, Juan C. Autinob, Gustavo P. Romanellib, c and Daniel O. Bennardi
European Journal of Medicinal Chemistry
Article in Press,

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http://dx.doi.org/10.1016/j.ejmech.2007.11.009

5. General Practitioners reduced benzodiazepine prescriptions in an intervention study: a multilevel application
Roy Stewarta, Wim J.M. Niessenb, Jan Broerb, Tom A.B. Snijdersc, Floor M. Haaijer-Ruskampd and Betty Meyboom-De Jong
Journal of Clinical Epidemiology
Volume 60, Issue 10, October 2007, Pages 1076.e1-1076.e10

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http://dx.doi.org/10.1016/j.jclinepi.2006.11.024

6. Robust fuzzy mappings for QSAR studies

Mohit Kumara, Kerstin Thurowa, , Norbert Stollb, and Regina Stoll
European Journal of Medicinal Chemistry
Volume 42, Issue 5, May 2007, Pages 675-685

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http://dx.doi.org/10.1016/j.ejmech.2006.12.017

7. A single point mutation of the GABAA receptor α5-subunit confers fluoxetine sensitivity
Jason M.C. Derry1, Isabelle M. Paulsena, Martin Daviesa and Susan M.J. Dunn
Neuropharmacology
Volume 52, Issue 2, February 2007, Pages 497-505

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http://dx.doi.org/10.1016/j.neuropharm.2006.07.036

8. PET imaging with [11C]PBR28 can localize and quantify upregulated peripheral benzodiazepine receptors associated with cerebral ischemia in rat

Masao Imaizumia, Hyun-Ju Kimb, Sami S. Zoghbia, Emmanuelle Briarda, Jinsoo Honga, John L. Musachioa, Christl Ruetzlerc, De-Maw Chuangb, Victor W. Pikea, Robert B. Innisa and Masahiro Fujita
Neuroscience Letters
Volume 411, Issue 3, 16 January 2007, Pages 200-205

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http://dx.doi.org/10.1016/j.neulet.2006.09.093

9. Synthesis, pharmacology and molecular modeling of N-substituted 2-phenyl-indoles and benzimidazoles as potent GABAA agonists
José Luis Falcó, Maria Piquéa, Miguel Gonzáleza, Irma Buiraa, Eva Méndeza, Jose Terencioa, Cristina Péreza, Marta Príncepa, Albert Palomera and Antonio Guglietta
European Journal of Medicinal Chemistry
Volume 41, Issue 8, August 2006, Pages 985-990

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http://dx.doi.org/10.1016/j.ejmech.2006.03.031

Заранее большое спасибо!

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[Ligand]

Да-а-а, литературка таки серьёёёзная.
Спасибо большое!